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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12910 | Sigma-1 receptor antagonist 1 | Sigma receptor | |
Sigma-1 receptor antagonist 1 is an effective and selective antagonist of sigma-1 receptor. Sigma-1 receptor antagonist 1 exhibits antineuropathic pain activity and can be used in the treatment of neuropathic pain studie... | |||
T12911 | Sigma-1 receptor antagonist 2 | Sigma receptor | |
Sigma-1 receptor antagonist 2 is a potent and selective antagonist of sigma 1 receptor (σ1 R) (σ1 and σ2 receptor with Kis of 3.88 and 1288 nM , respectively). | |||
T12912 | Sigma-1 receptor antagonist 3 | Sigma receptor , HER | |
Sigma-1 receptor antagonist 3 is a potent and selective antagonist of Sigma-1 (σ1) receptor(Ki : 1.14 nM), has the potential for the neuropathic pain. | |||
T16883 | Sigma-2 receptor antagonist 1 | Others | |
Sigma-2 receptor antagonist 1 is an antagonist of the sigma-2 (σ-2) receptor. | |||
T22870 | IPAG | Opioid Receptor | |
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis. | |||
T21788 | BD 1008 dihydrobromide | Sigma receptor | |
BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors. | |||
T5389 | Volinanserin | M 100907,MDL100907 | 5-HT Receptor |
Volinanserin (MDL100907) (MDL 100907) is a potent and selective antagonist of the serotonin receptor 5-HT2 (Ki: 0.36 nM) and shows 300-fold selectivity for 5-HT2 receptor over 5-HT1c, alpha-1 adrenergic and sigma recepto... | |||
T61901 | σ1 Receptor/μ Opioid receptor modulator 1 | ||
σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM). Opioid receptor modulator 1 shows potent analgesic activity, and ... |